Development and evaluation of a vaginal ring device for sustained delivery of HIV microbicides to non-human primates

J Med Primatol. 2009 Aug;38(4):263-71. doi: 10.1111/j.1600-0684.2009.00354.x. Epub 2009 May 19.

Abstract

Background: There is considerable interest in developing coitally independent, sustained release formulations for long-term administration of HIV microbicides. Vaginal ring devices are at the forefront of this formulation strategy.

Methods: Non-medicated silicone elastomer vaginal rings were prepared having a range of appropriate dimensions for testing vaginal fit in pig-tailed and Chinese rhesus macaques. Cervicovaginal proinflammatory markers were evaluated. Compression testing was performed to compare the relative flexibility of various macaque and commercial human rings.

Results: All rings remained in place during the study period and no tissue irritation or significant induction of cervicovaginal proinflammatory markers or signs of physical discomfort were observed during the 8-week study period.

Conclusions: Qualitative evaluation suggests that the 25 x 5-mm ring provided optimal fit in both macaque species. Based on the results presented here, low-consistency silicone elastomers do not cause irritation in macaques and are proposed as suitable materials for the manufacture of microbicide-loaded vaginal rings.

MeSH terms

  • Administration, Intravaginal
  • Animals
  • Anti-HIV Agents / administration & dosage*
  • Equipment and Supplies* / adverse effects
  • Equipment and Supplies* / veterinary
  • Female
  • HIV
  • Macaca mulatta
  • Macaca nemestrina
  • Mechanics

Substances

  • Anti-HIV Agents