Androgen receptor regulates a distinct transcription program in androgen-independent prostate cancer

Cell. 2009 Jul 23;138(2):245-56. doi: 10.1016/j.cell.2009.04.056.

Abstract

The evolution of prostate cancer from an androgen-dependent state to one that is androgen-independent marks its lethal progression. The androgen receptor (AR) is essential in both, though its function in androgen-independent cancers is poorly understood. We have defined the direct AR-dependent target genes in both androgen-dependent and -independent cancer cells by generating AR-dependent gene expression profiles and AR cistromes. In contrast to what is found in androgen-dependent cells, AR selectively upregulates M-phase cell-cycle genes in androgen-independent cells, including UBE2C, a gene that inactivates the M-phase checkpoint. We find that epigenetic marks at the UBE2C enhancer, notably histone H3K4 methylation and FoxA1 transcription factor binding, are present in androgen-independent cells and direct AR-enhancer binding and UBE2C activation. Thus, the role of AR in androgen-independent cancer cells is not to direct the androgen-dependent gene expression program without androgen, but rather to execute a distinct program resulting in androgen-independent growth.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Androgens / metabolism
  • Cell Division
  • Cell Line, Tumor
  • Gene Expression Regulation, Neoplastic*
  • Hepatocyte Nuclear Factor 3-alpha / metabolism
  • Histones / metabolism
  • Humans
  • Male
  • Prostatic Neoplasms / genetics
  • Prostatic Neoplasms / metabolism*
  • Receptors, Androgen / metabolism*
  • Transcriptional Activation
  • Ubiquitin-Conjugating Enzymes / metabolism

Substances

  • AR protein, human
  • Androgens
  • FOXA1 protein, human
  • Hepatocyte Nuclear Factor 3-alpha
  • Histones
  • Receptors, Androgen
  • UBE2C protein, human
  • Ubiquitin-Conjugating Enzymes