Comparison of the central and renal dopamine-1 receptor

Am J Hypertens. 1990 Jun;3(6 Pt 2):37S-39S. doi: 10.1093/ajh/3.6.37s.

Abstract

The dopamine D-1 receptor from striatal membranes was compared with the dopamine DA-1 receptor from renal proximal tubules. The dopamine-1 receptors were solubilized with 1% sodium cholate and phospholipids after pretreatment with the dopamine-1 agonist, SKF R-38393. The soluble receptors were reconstituted into phospholipid vesicles after removal of sodium cholate. The receptors were studied by radioligand binding using the dopamine-1 antagonist [125I]-SCH 23982. The reconstituted dopamine D-1 and DA-1 receptor densities were similar. However, the affinity of the solubilized D-1 receptor was 17-fold greater than the solubilized DA-1 receptor. The affinity of membrane bound D-1 receptor to the radioligand was also greater than that noted for membrane bound DA-1 receptor. The mechanism for this difference remains to be determined.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine / metabolism
  • Affinity Labels
  • Animals
  • Benzazepines* / analogs & derivatives*
  • Benzazepines* / metabolism
  • Binding, Competitive
  • Corpus Striatum / metabolism*
  • Dopamine Agents / metabolism
  • Kidney Tubules, Proximal / metabolism*
  • Rats
  • Receptors, Dopamine / metabolism*
  • Receptors, Dopamine D1
  • Solubility

Substances

  • 8-iodo-2,3,4,5-tetrahydro-3-methyl-5-phenyl-1H-3-benzazepine-7-ol
  • Affinity Labels
  • Benzazepines
  • Dopamine Agents
  • Receptors, Dopamine
  • Receptors, Dopamine D1
  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine