Normal responsiveness of superficial hand veins to alpha- and beta-adrenergic stimuli in allergic asthma: effects of terbutaline and prednisolone on beta-adrenergic responsiveness

J Allergy Clin Immunol. 1990 Nov;86(5):714-25. doi: 10.1016/s0091-6749(05)80175-7.

Abstract

Impaired function of the adrenergic-receptor system has been postulated to contribute to the pathogenesis of bronchial asthma. Using the dorsal hand-vein compliance technique, we compared the changes in diameter of superficial hand veins in response to phenylephrine, an alpha-adrenoceptor agonist, and to isoproterenol, a beta-adrenoceptor agonist, in 14 untreated patients with allergic asthma and in 16 nonatopic control subjects. There were no significant differences in the median effective dose of phenylephrine that produced 50% of maximal venoconstriction (ED50) or in the maximal response (Emax) between the two groups. Bronchial hyperreactivity (assessed by methacholine-challenge tests) in the patients with asthma was uncorrelated with the ED50 or Emax of isoproterenol. These results demonstrate no evidence for a generalized change in alpha- or beta-adrenergic responsiveness on smooth muscle cells in asthma. Hand-vein responsiveness to isoproterenol was unchanged after treatment for 7 days with oral terbutaline (5 mg three times per day). Thus, unlike leukocytes, smooth muscle appears not readily susceptible to beta-adrenoceptor desensitization in vivo. Local infusions of prednisolone or dexamethasone during 2 hours and systemic administration of dexamethasone (24 hours) caused a significant fall in the Emax for isoproterenol. The mechanism of attenuation of beta-adrenoceptor responsiveness by corticosteroids remains to be determined.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adrenergic alpha-Antagonists / pharmacology*
  • Adrenergic beta-Antagonists / pharmacology*
  • Adult
  • Analysis of Variance
  • Asthma / physiopathology*
  • Dose-Response Relationship, Drug
  • Forced Expiratory Volume / drug effects
  • Hand / blood supply
  • Humans
  • Isoproterenol / pharmacology
  • Male
  • Methacholine Compounds / administration & dosage
  • Phenylephrine / pharmacology
  • Prednisolone / pharmacology*
  • Receptors, Adrenergic, alpha / drug effects*
  • Terbutaline / pharmacology*
  • Vasoconstriction / drug effects

Substances

  • Adrenergic alpha-Antagonists
  • Adrenergic beta-Antagonists
  • Methacholine Compounds
  • Receptors, Adrenergic, alpha
  • Phenylephrine
  • Prednisolone
  • Isoproterenol
  • Terbutaline