32P-postlabeling of N-7, N2 and O6 2'-deoxyguanosine 3'-monophosphate adducts of styrene oxide

Chem Biol Interact. 1991;77(1):39-50. doi: 10.1016/0009-2797(91)90004-q.

Abstract

Adducts were prepared by reacting styrene oxide with 2-deoxyguanosine 3'-monophosphate (dGMP). Four isomeric N-7-, two diastereomeric N2- and three isomeric O6-adduct were isolated and characterized. The adducts were used as substrates in the 32P-postlabeling reaction. No phosphorylation products were seen with the N-7-alkylation products. One diastereomeric N2-adduct was labeled with 20% efficiency and the second with a markedly lower efficiency. Two of the three O6-adducts were labeled with 5% and the third with 10% labeling efficiency. The results suggest that large N-7-dGMP adducts are very poor substrates of T4 polynucleotide kinase. The diastereomeric products are labeled at different efficiencies indicating stereoselectivity in the kinase reaction.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Deoxyguanine Nucleotides*
  • Epoxy Compounds*
  • Phosphorus Radioisotopes
  • Phosphorylation
  • Polynucleotide 5'-Hydroxyl-Kinase / pharmacology
  • Stereoisomerism

Substances

  • Deoxyguanine Nucleotides
  • Epoxy Compounds
  • Phosphorus Radioisotopes
  • 2'-deoxyguanosine 5'-phosphate
  • styrene oxide
  • Polynucleotide 5'-Hydroxyl-Kinase