Total syntheses of isodomoic acids G and H: an exercise in tetrasubstituted alkene synthesis

J Am Chem Soc. 2009 Dec 9;131(48):17714-8. doi: 10.1021/ja907931u.

Abstract

A unified approach to the pyrrolidine triacid natural products isodomoic acids G and H has been developed. Total syntheses of both natural products were completed, and determination of the correct stereostructure of isodomoic acid G was established by comparing 5'-(R) and 5'-(S) isomers to a sample of authentic material. A nickel-catalyzed cyclization constructs the pyrrolidine ring while simultaneously establishing either the E or Z stereochemistry of an exocyclic tetrasubstituted alkene. Stereoselective assembly of both the E- and Z-alkenes of the natural products is made possible by a predictable strategy that alters the timing of substituent introduction to control alkene stereochemistry.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Alkenes / chemical synthesis*
  • Alkenes / chemistry*
  • Biological Products / chemical synthesis
  • Biological Products / chemistry
  • Cyclization
  • Heptanoic Acids / chemical synthesis*
  • Heptanoic Acids / chemistry
  • Stereoisomerism
  • Substrate Specificity

Substances

  • Alkenes
  • Biological Products
  • Heptanoic Acids
  • isodomoic acid G
  • isodomoic acid H