Abstract
Prostaglandins (PGs) have been shown to inhibit tumour metastases in experimental animal systems. Nafazatrom is a pyrazolinone derivative that increases endogenous prostacyclin (PGI2) and has experimental anti-cancer activity. In the present study, nafazatrom was given to 47 women with advanced breast cancer; objective remission of metastases was seen in 2 patients and stabilisation of disease in 1 case. Nafazatrom was safe and well tolerated.
MeSH terms
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Aged
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Antineoplastic Agents / adverse effects
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Antineoplastic Agents / pharmacology
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Antineoplastic Agents / therapeutic use*
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Breast Neoplasms / drug therapy*
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Breast Neoplasms / pathology
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Drug Evaluation
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Female
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Humans
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Middle Aged
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Prostaglandins / biosynthesis
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Pyrazoles / adverse effects
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Pyrazoles / pharmacology
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Pyrazoles / therapeutic use*
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Pyrazolones*
Substances
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Antineoplastic Agents
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Prostaglandins
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Pyrazoles
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Pyrazolones
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nafazatrom