Stress and GABA receptors

J Neurochem. 2010 Mar;112(5):1115-30. doi: 10.1111/j.1471-4159.2009.06539.x. Epub 2009 Dec 10.

Abstract

GABA(A) receptors are sensitive to subtle changes in the environment in both early-life and adulthood. These neurochemical responses to stress in adulthood are sex-dependent. Acute stress induces rapid changes in GABA(A) receptors in experimental animals, with the direction of the changes varying according to the sex of the animals and the stress-paradigm studied. These rapid alterations are of particular interest as they provide an example of fast neurotransmitter system plasticity that may be mediated by stress-induced increases in neurosteroids, perhaps via effects on phosphorylation and/or receptor trafficking. Interestingly, some studies have also provided evidence for long-lasting changes in GABA(A) receptors as a result of exposure to stressors in early-life. The short- and long-term stress sensitivity of the GABAergic system implicates GABA(A) receptors in the non-genetic etiology of psychiatric illnesses such as depression and schizophrenia in which stress may be an important factor.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Allosteric Site
  • Animals
  • GABA Agents / pharmacology
  • Humans
  • Models, Animal
  • Phosphorylation
  • Protein Transport / physiology
  • Receptors, GABA / genetics
  • Receptors, GABA / metabolism*
  • Sex Factors
  • Stress, Psychological / genetics
  • Stress, Psychological / metabolism*

Substances

  • GABA Agents
  • Receptors, GABA