About the mutagenicity of chlorine-substituted furanones and halopropenals. A QSAR study using molecular orbital indices

Mutat Res. 1991 Mar;247(1):97-102. doi: 10.1016/0027-5107(91)90037-o.

Abstract

Electron affinities, frontier molecular orbital energies and electron densities at individual carbon atoms were calculated for 11 chlorofuranones including the strong mutagen 3-chloro-4-(dichloromethyl)-5-hydroxy-2(5H)-furanone (MX) and for 5 halopropenals by semi-empirical AM1 and ab initio STO-3G methods. Significant correlations were found between Ames TA100 mutagenicity and the following AM1 electronic parameters of chlorofuranones: electron affinity (r = 0.9556). LUMO energy (r = 0.9332) and frontier electron density of LUMO at the alpha-carbon (r = 0.8882). In halopropenals only LUMO electron density at the beta-carbon correlates well with mutagenicity. The observed correlations suggest a reaction mechanism in which chlorofuranones and halopropenals act as electron acceptors in the interaction with DNA.

MeSH terms

  • Aldehydes / chemistry
  • Aldehydes / toxicity*
  • Alkenes / chemistry
  • Alkenes / toxicity*
  • Chlorine / chemistry*
  • Furans / chemistry
  • Furans / toxicity*
  • Halogens / chemistry
  • Halogens / toxicity
  • Molecular Structure
  • Mutagenicity Tests
  • Mutagens / chemistry
  • Mutagens / toxicity*
  • Salmonella typhimurium / genetics

Substances

  • Aldehydes
  • Alkenes
  • Furans
  • Halogens
  • Mutagens
  • Chlorine