GADD45beta enhances Col10a1 transcription via the MTK1/MKK3/6/p38 axis and activation of C/EBPbeta-TAD4 in terminally differentiating chondrocytes

J Biol Chem. 2010 Mar 12;285(11):8395-407. doi: 10.1074/jbc.M109.038638. Epub 2010 Jan 4.

Abstract

GADD45beta (growth arrest- and DNA damage-inducible) interacts with upstream regulators of the JNK and p38 stress response kinases. Previously, we reported that the hypertrophic zone of the Gadd45beta(-/-) mouse embryonic growth plate is compressed, and expression of type X collagen (Col10a1) and matrix metalloproteinase 13 (Mmp13) genes is decreased. Herein, we report that GADD45beta enhances activity of the proximal Col10a1 promoter, which contains evolutionarily conserved AP-1, cAMP-response element, and C/EBP half-sites, in synergism with C/EBP family members, whereas the MMP13 promoter responds to GADD45beta together with AP-1, ATF, or C/EBP family members. C/EBPbeta expression also predominantly co-localizes with GADD45beta in the embryonic growth plate. Moreover, GADD45beta enhances C/EBPbeta activation via MTK1, MKK3, and MKK6, and dominant-negative p38alphaapf, but not JNKapf, disrupts the combined trans-activating effect of GADD45beta and C/EBPbeta on the Col10a1 promoter. Importantly, GADD45beta knockdown prevents p38 phosphorylation while decreasing Col10a1 mRNA levels but does not affect C/EBPbeta binding to the Col10a1 promoter in vivo, indicating that GADD45beta influences the transactivation function of DNA-bound C/EBPbeta. In support of this conclusion, we show that the evolutionarily conserved TAD4 domain of C/EBPbeta is the target of the GADD45beta-dependent signaling. Collectively, we have uncovered a novel molecular mechanism linking GADD45beta via the MTK1/MKK3/6/p38 axis to C/EBPbeta-TAD4 activation of Col10a1 transcription in terminally differentiating chondrocytes.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Activating Transcription Factor 1 / metabolism
  • Animals
  • Antigens, Differentiation / metabolism*
  • CCAAT-Enhancer-Binding Protein-beta / metabolism*
  • Cell Differentiation / physiology
  • Cell Line, Tumor
  • Chondrocytes / cytology*
  • Chondrocytes / physiology*
  • Collagen Type X / genetics*
  • Cyclic AMP Response Element-Binding Protein / metabolism
  • Gene Expression Regulation, Developmental
  • Growth Plate / cytology
  • Growth Plate / embryology
  • Growth Plate / physiology
  • Humans
  • MAP Kinase Kinase 3 / metabolism
  • MAP Kinase Kinase 6 / metabolism
  • MAP Kinase Kinase Kinase 1 / metabolism
  • MAP Kinase Kinase Kinase 4 / metabolism
  • MAP Kinase Signaling System / physiology*
  • Matrix Metalloproteinase 13 / genetics
  • Mice
  • Mice, Inbred C57BL
  • Promoter Regions, Genetic / physiology
  • Teratocarcinoma
  • Transcription Factor AP-1 / metabolism
  • Transcription, Genetic / physiology
  • p38 Mitogen-Activated Protein Kinases / metabolism

Substances

  • Activating Transcription Factor 1
  • Antigens, Differentiation
  • Atf1 protein, mouse
  • CCAAT-Enhancer-Binding Protein-beta
  • Cebpb protein, mouse
  • Collagen Type X
  • Creb1 protein, mouse
  • Cyclic AMP Response Element-Binding Protein
  • Gadd45b protein, mouse
  • Transcription Factor AP-1
  • p38 Mitogen-Activated Protein Kinases
  • MAP Kinase Kinase Kinase 1
  • MAP Kinase Kinase Kinase 4
  • MAP Kinase Kinase 3
  • MAP Kinase Kinase 6
  • Map2k3 protein, mouse
  • Map2k6 protein, mouse
  • Matrix Metalloproteinase 13
  • Mmp13 protein, mouse