Assembly and stoichiometry of the AMPA receptor and transmembrane AMPA receptor regulatory protein complex

J Neurosci. 2010 Jan 20;30(3):1064-72. doi: 10.1523/JNEUROSCI.3909-09.2010.

Abstract

Glutamate is a major excitatory neurotransmitter in the vertebrate brain. AMPA-type glutamate receptors mediate fast excitatory transmission. AMPA receptors assemble with transmembrane AMPA receptor regulatory protein (TARP) auxiliary subunits and function as native ion channels. However, the assembly and stoichiometry of AMPA receptor and TARP complexes remain unclear. Here, we developed a novel strategy to determine the assembly and stoichiometry of this protein complex and found that functional AMPA receptors indeed assembled as a tetramer in a dimer-of-dimers structure. Furthermore, we found that the AMPA receptor auxiliary subunit, TARP, had a variable stoichiometry (1-4 TARP units) on AMPA receptors and that 1 TARP unit was sufficient to modulate AMPA receptor activity. In neurons, TARP had fixed and minimum stoichiometry on AMPA receptors. This fundamental composition of the AMPA receptor/TARP complex is important for the elucidation of the molecular machinery that underlies synaptic transmission.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium Channels / genetics
  • Calcium Channels / metabolism
  • Green Fluorescent Proteins / genetics
  • Hemagglutinins / metabolism
  • Larva
  • Membrane Potentials / drug effects
  • Membrane Potentials / genetics
  • Models, Molecular
  • Mutation / genetics
  • Nuclear Proteins / metabolism*
  • Oocytes
  • Patch-Clamp Techniques
  • Protein Conformation
  • Receptors, AMPA / genetics
  • Receptors, AMPA / metabolism*
  • Receptors, Glutamate / genetics
  • Stochastic Processes
  • Transcription, Genetic
  • Xenopus
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid / pharmacology

Substances

  • Cacng2 protein, rat
  • Calcium Channels
  • Hemagglutinins
  • Nuclear Proteins
  • Receptors, AMPA
  • Receptors, Glutamate
  • TARP
  • Green Fluorescent Proteins
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
  • glutamate receptor ionotropic, AMPA 1