Cholecystokinin-A receptor mediation of food intake in cats

Am J Physiol. 1991 Apr;260(4 Pt 2):R693-7. doi: 10.1152/ajpregu.1991.260.4.R693.

Abstract

The selective cholecystokinin (CCK)-B-receptor agonist and antagonist, BC 264 and L 365260, respectively, and the CCK-A-receptor antagonist, L 364718, were used to investigate the possible involvement of different classes of CCK receptors in the control of food intake induced by exogenous CCK octapeptide (CCK-8) in the cat with gastric fistula. Intravenous infusion of CCK-8 dose dependently inhibited milk intake under sham-feeding conditions, maximal inhibition reaching 52 +/- 7% (P less than 0.001) with 0.88 nmol.kg-1.h-1. L 364718 prevented this inhibition, whereas L 365260 was ineffective over the dose range tested. The reversal effect of L 364718 on 0.88 nmol.kg-1.h-1 CCK-8-induced inhibition of milk intake was observed at doses as low as 0.44 nmol.kg-1.h-1. The selective CCK-B-receptor agonist, BC 264, in doses ranging from 0.88 to 7 nmol.kg-1.h-1, had no effect on milk intake under sham-feeding conditions, although it dose dependently stimulated gastric acid output. Furthermore, neither L 364718 nor L 365260 (88 nmol.kg-1.h-1 iv) stimulated milk intake when given in the absence of CCK-8. We conclude that exogenous CCK-8 causes satiety in the cat through activation of peripheral CCK-A receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzodiazepinones / administration & dosage
  • Benzodiazepinones / pharmacology
  • Cats
  • Cholecystokinin / administration & dosage
  • Cholecystokinin / analogs & derivatives
  • Cholecystokinin / pharmacology
  • Devazepide
  • Dose-Response Relationship, Drug
  • Eating / drug effects
  • Eating / physiology*
  • Gastric Acid / metabolism
  • Milk
  • Peptide Fragments / administration & dosage
  • Peptide Fragments / pharmacology
  • Phenylurea Compounds*
  • Receptors, Cholecystokinin / antagonists & inhibitors
  • Receptors, Cholecystokinin / physiology*
  • Satiation / drug effects
  • Satiation / physiology
  • Sincalide / pharmacology

Substances

  • BC 264
  • Benzodiazepinones
  • Peptide Fragments
  • Phenylurea Compounds
  • Receptors, Cholecystokinin
  • L 365260
  • Cholecystokinin
  • Devazepide
  • Sincalide