Metabolism of almitrine in extensive and poor metabolisers of debrisoquine/sparteine

Br J Clin Pharmacol. 1991 Jan;31(1):73-6. doi: 10.1111/j.1365-2125.1991.tb03859.x.

Abstract

1. Almitrine bismesylate displays wide inter-subject variation in peak plasma concentrations and can induce peripheral polyneuropathy. 2. The phenotyped volunteer panel approach was used to examine whether almitrine oxidation displayed a genetic polymorphism of the debrisoquine/sparteine type. 3. There was no difference between poor and extensive metabolisers of debrisoquine with respect to the pharmacokinetics and metabolism of almitrine.

MeSH terms

  • Adult
  • Almitrine / metabolism*
  • Chromatography, High Pressure Liquid
  • Debrisoquin / metabolism*
  • Female
  • Humans
  • Male
  • Oxidation-Reduction
  • Phenotype
  • Polymorphism, Genetic
  • Sparteine / metabolism*

Substances

  • Sparteine
  • Almitrine
  • Debrisoquin