MYCN oncoprotein targets and their therapeutic potential

Cancer Lett. 2010 Jul 28;293(2):144-57. doi: 10.1016/j.canlet.2010.01.015. Epub 2010 Feb 13.

Abstract

The MYCN oncogene encodes a transcription factor which is amplified in up to 40% of high risk neuroblastomas. MYCN amplification is a well-established poor prognostic marker in neuroblastoma, however the role of MYCN expression and the mechanisms by which it acts to promote an aggressive phenotype remain largely unknown. This review discusses the current evidence identifying the direct and indirect downstream transcriptional targets of MYCN from recent studies, with particular reference to how MYCN affects the cell cycle, DNA damage response, differentiation and apoptosis in neuroblastoma.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Apoptosis / genetics
  • Brain Neoplasms / genetics*
  • Brain Neoplasms / therapy
  • Cell Cycle / genetics
  • Cell Differentiation / genetics
  • Cell Line, Tumor
  • DNA Damage
  • Drug Delivery Systems*
  • Gene Expression Profiling
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Immunoglobulin G / therapeutic use
  • Melphalan / therapeutic use
  • N-Myc Proto-Oncogene Protein
  • Neuroblastoma / genetics*
  • Neuroblastoma / therapy
  • Nuclear Proteins / genetics*
  • Oncogene Proteins / genetics*
  • Transcription Factors / genetics*

Substances

  • Immunoglobulin G
  • MYCN protein, human
  • N-Myc Proto-Oncogene Protein
  • Nuclear Proteins
  • Oncogene Proteins
  • Transcription Factors
  • antineoplastic agent K 18
  • Melphalan