Abstract
Objective:
Atherosclerosis is an inflammatory disease. Autoimmune responses to low-density lipoproteins (LDL) contribute to its progression, whereas immunization with LDL may induce atheroprotective or proatherogenic responses. The objective of this study was to develop an atheroprotective vaccine by targeting a peptide of the LDL protein constituent apolipoprotein B-100 (apoB-100) to the nasal mucosa to induce a protective mucosal immune response.
Methods and results:
A peptide comprising amino acids 3136 to 3155 of apoB-100 (p210) was fused to the B subunit of cholera toxin (CTB), which binds to a ganglioside on mucosal epithelia. The effect of nasal administration of the p210-CTB fusion protein on atherogenesis was compared with that of an ovalbumin peptide fused to CTB and with untreated controls. Immunization with p210-CTB for 12 weeks caused a 35% reduction in aortic lesion size in Apoe(-/-) mice. This effect was accompanied by induction of regulatory T cells that markedly suppressed effector T cells rechallenged with apoB-100 and increased numbers of interleukin (IL)-10(+) CD4(+) T cells. Furthermore, a peptide-specific antibody response was observed. Atheroprotection was also documented in apoe(-/-) mice lacking functional transforming growth factor-beta receptors on T cells.
Conclusion:
Nasal administration of an apoB-100 peptide fused to CTB attenuates atherosclerosis and induces regulatory Tr1 cells that inhibit T effector responses to apoB-100.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Administration, Intranasal
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Aerosols
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Animals
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Aortic Diseases / genetics
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Aortic Diseases / immunology
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Aortic Diseases / metabolism
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Aortic Diseases / pathology
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Aortic Diseases / prevention & control*
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Apolipoprotein B-100 / administration & dosage*
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Apolipoprotein B-100 / immunology
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Apolipoproteins E / deficiency
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Apolipoproteins E / genetics
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Atherosclerosis / genetics
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Atherosclerosis / immunology
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Atherosclerosis / metabolism
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Atherosclerosis / pathology
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Atherosclerosis / prevention & control*
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Cholera Toxin / administration & dosage*
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Cholera Toxin / immunology
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Disease Models, Animal
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Female
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Forkhead Transcription Factors / genetics
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Humans
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Immunity, Cellular / drug effects
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Immunity, Humoral / drug effects
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Immunity, Mucosal / drug effects
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Immunoconjugates / administration & dosage*
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Immunoconjugates / immunology
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Interleukin-10 / genetics
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Mice
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Mice, Knockout
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Nasal Mucosa / drug effects
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Nasal Mucosa / immunology
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Ovalbumin / administration & dosage
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Ovalbumin / immunology
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Peptide Fragments / administration & dosage*
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Peptide Fragments / immunology
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Protein Serine-Threonine Kinases / metabolism
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RNA, Messenger / metabolism
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Receptor, Transforming Growth Factor-beta Type II
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Receptors, Transforming Growth Factor beta / metabolism
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T-Lymphocytes, Regulatory / drug effects*
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T-Lymphocytes, Regulatory / immunology
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Vaccines, Synthetic / administration & dosage*
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Vaccines, Synthetic / immunology
Substances
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Aerosols
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Apolipoprotein B-100
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Apolipoproteins E
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Forkhead Transcription Factors
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Foxp3 protein, mouse
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Immunoconjugates
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Peptide Fragments
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RNA, Messenger
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Receptors, Transforming Growth Factor beta
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Vaccines, Synthetic
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Interleukin-10
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Ovalbumin
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Cholera Toxin
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Protein Serine-Threonine Kinases
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Receptor, Transforming Growth Factor-beta Type II