Contrasting behavior of conformationally locked carbocyclic nucleosides of adenosine and cytidine as substrates for deaminases

Nucleosides Nucleotides Nucleic Acids. 2009 May;28(5):614-32. doi: 10.1080/15257770903091904.

Abstract

In addition to the already known differences between adenosine deaminase (ADA) and cytidine deaminase (CDA) in terms of their tertiary structure, the sphere of Zn(+2) coordination, and their reverse stereochemical preference, we present evidence that the enzymes also differ significantly in terms of the North/South conformational preferences for their substrates and the extent to which the lack of the O(4') oxygen affects the kinetics of the enzymatic deamination of carbocyclic substrates. The carbocyclic nucleoside substrates used in this study have either a flexible cyclopentane ring or a rigid bicyclo[3.1.0]hexane scaffold.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adenosine / chemistry*
  • Adenosine / metabolism
  • Adenosine Deaminase / chemistry
  • Adenosine Deaminase / metabolism*
  • Animals
  • Cattle
  • Cytidine / chemistry*
  • Cytidine / metabolism
  • Cytidine Deaminase / chemistry
  • Cytidine Deaminase / metabolism*
  • Models, Molecular
  • Molecular Conformation

Substances

  • Cytidine
  • Adenosine Deaminase
  • Cytidine Deaminase
  • Adenosine