Interaction of connexin43 and protein kinase C-delta during FGF2 signaling

BMC Biochem. 2010 Mar 25:11:14. doi: 10.1186/1471-2091-11-14.

Abstract

Background: We have recently demonstrated that modulation of the gap junction protein, connexin43, can affect the response of osteoblasts to fibroblast growth factor 2 in a protein kinase C-delta-dependent manner. Others have shown that the C-terminal tail of connexin43 serves as a docking platform for signaling complexes. It is unknown whether protein kinase C-delta can physically interact with connexin43.

Results: In the present study, we investigate by immunofluorescent co-detection and biochemical examination the interaction between Cx43 and protein kinase C-delta. We establish that protein kinase C-delta physically interacts with connexin43 during fibroblast growth factor 2 signaling, and that protein kinase C delta preferentially co-precipitates phosphorylated connexin43. Further, we show by pull down assay that protein kinase C-delta associates with the C-terminal tail of connexin43.

Conclusions: Connexin43 can serve as a direct docking platform for the recruitment of protein kinase C-delta in order to affect fibroblast growth factor 2 signaling in osteoblasts. These data expand the list of signal molecules that assemble on the connexin43 C-terminal tail and provide a critical context to understand how gap junctions modify signal transduction cascades in order to impact cell function.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Connexin 43 / metabolism*
  • Fibroblast Growth Factor 2 / metabolism*
  • Immunoprecipitation
  • Osteoblasts / metabolism
  • Phosphorylation
  • Protein Interaction Domains and Motifs
  • Protein Kinase C-delta / metabolism*
  • Signal Transduction*

Substances

  • Connexin 43
  • GJA1 protein, mouse
  • Fibroblast Growth Factor 2
  • Protein Kinase C-delta