Microbial metabolism. Part 11. Metabolites of flutamide

Chem Pharm Bull (Tokyo). 2010 Apr;58(4):562-4. doi: 10.1248/cpb.58.562.

Abstract

The yeast culture, Rhodotorula mucilaginosa (ATCC 20129) transformed flutamide (1) to three metabolites: 4-nitro-3-(trifluoromethyl)aniline (2), 2-methyl-N-[4-amino-3-(trifloromethyl)phenyl]propanamide (3) and N-[4-amino-3-(trifluoromethyl)phenyl]acetamide (4). The structures were established by spectroscopic methods.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Antineoplastic Agents, Hormonal / chemistry
  • Antineoplastic Agents, Hormonal / metabolism*
  • Flutamide / chemistry
  • Flutamide / metabolism*
  • Humans
  • Molecular Structure
  • Rhodotorula / chemistry
  • Rhodotorula / metabolism*

Substances

  • Antineoplastic Agents, Hormonal
  • Flutamide