The uremic solute indoxyl sulfate acts as an antioxidant against superoxide anion radicals under normal-physiological conditions

FEBS Lett. 2010 Jul 2;584(13):2816-20. doi: 10.1016/j.febslet.2010.04.046. Epub 2010 Apr 21.

Abstract

The effect of the uremic solute indoxyl sulfate (IS) on scavenging superoxide anion radicals (O(2)(*-)) generated from both the xanthine/xanthine oxidase (X/XO) system and activated neutrophils was investigated by electron paramagnetic resonance spectroscopy, combined with 2-ethoxycarbonyl-2-methyl-3,4-dihydro-2H-pyrrole-1-oxide (EMPO). The findings show that the presence of normal-physiological serum concentrations of IS (0.1-10 microM) resulted in decreased formation of EMPO-superoxide adduct without affecting XO activity. Furthermore, IS showed scavenging activity against cell-derived O(2)(*-) generated from activated neutrophils. In addition, IS also eliminated hydroxyl radicals. These findings suggest that IS acts as a novel endogenous antioxidant under normal-physiological conditions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antioxidants / chemistry*
  • Electron Spin Resonance Spectroscopy
  • Humans
  • Indican / blood
  • Indican / chemistry*
  • Neutrophils / metabolism
  • Pyrroles / chemistry
  • Superoxides / chemistry*

Substances

  • 2-ethoxycarbonyl-2-methyl-3,4-dihydro-2H-pyrrole-1-oxide
  • Antioxidants
  • Pyrroles
  • Superoxides
  • Indican