Synthesis of pyrazolines by a site isolated resin-bound reagents methodology

Org Biomol Chem. 2010 Jul 21;8(14):3287-93. doi: 10.1039/c004704j. Epub 2010 May 26.

Abstract

The elaboration of biologically important 3,4-substituted pyrazolines was achieved by an organocatalysed aza-Michael/transimination domino sequence between hydrazones and enones making use of a mixture of heterogeneous resin-bound acid/base reagents. This methodology nicely illustrates the site isolation concept of supported reagents allowing the simultaneous use of otherwise destructive reactive functionalities.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Catalysis
  • Hydrogen-Ion Concentration
  • Indicators and Reagents / chemistry
  • Pyrazoles / chemical synthesis*
  • Pyrazoles / chemistry*
  • Resins, Synthetic / chemistry*

Substances

  • Indicators and Reagents
  • Pyrazoles
  • Resins, Synthetic
  • pyrazole