TargetScreen: an unbiased approach to identify functionally important microRNA targets

Cell Cycle. 2010 Jun 1;9(11):2080-4. doi: 10.4161/cc.9.11.11807. Epub 2010 Jun 1.

Abstract

We recently identified miR-19 as the critical activity for leukemogenesis within the oncogenic 17~92 cluster of microRNAs. ( 1) This finding prompted us to test an unbiased method for pinpointing those miR-19 targets may be key to its oncogenic action. Specifically, we used a large-scale short hairpin RNA screen to identify those miR-19 target genes, whose knockdown could reproduce miR-19's effects on lymphocyte transformation. In this way, we found that miR-19 produces a coordinate clampdown on multiple negative regulators of PI3K-related survival signals. These findings have implications for the therapy of miR-19 expressing tumors. They also validate a new strategy for the unbiased identification of functionally important microRNA target genes. Using the example of miR-19 in leukemia, we will discuss some possibilities and limitations of this new approach.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Gene Expression Regulation, Neoplastic*
  • Gene Knockdown Techniques
  • Humans
  • Leukemia / genetics*
  • Leukemia / therapy
  • MicroRNAs / antagonists & inhibitors
  • MicroRNAs / metabolism*
  • Phosphatidylinositol 3-Kinases / metabolism
  • RNA Interference

Substances

  • MIRN19 microRNA, human
  • MicroRNAs
  • Phosphatidylinositol 3-Kinases