The pentapeptide PLNPK inhibits systemic lupus erythematosus-associated renal damage

Inflamm Res. 2010 Dec;59(12):1081-9. doi: 10.1007/s00011-010-0228-y. Epub 2010 Jul 1.

Abstract

Objective: This study aimed to observe the therapeutic effect of pentapeptide PLNPK on systemic lupus erythematosus (SLE) in mice, and to study the inhibitory effect of PLNPK on activation of T cells in vivo.

Methods: Murine SLE-like chronic graft-versus-host disease (cGVHD) was induced. After treatment with PLNPK (100, 200, 400 μg/kg per day) for 70 days, serum blood urea nitrogen, creatine, total cholesterol, triglyceride and albumin were tested, and serum levels of anti-dsDNA and anti-histone antibodies were detected by ELISA. The pathological damage and IgG deposition in the kidney were identified. Concanavalin A (ConA)-induced T lymphocyte proliferation in SLE mice was also tested.

Results: PLNPK can reduce serum blood urea nitrogen, creatine, total cholesterol, triglyceride, and elevate serum albumin, and reduce levels of anti-dsDNA and anti-histone antibodies in the murine SLE model. Pathological damage and IgG deposition in the kidney were reduced in the PLNPK-treated group. PLNPK inhibited T lymphocyte infiltration in kidney tissues and ConA-induced T lymphocyte proliferation in SLE mice.

Conclusion: Our results demonstrate that PLNPK can suppress T cell function and reduce the production of autoantibodies, and may be a feasible and effective therapy in the SLE model.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Autoantibodies / immunology
  • Disease Models, Animal
  • Female
  • Graft vs Host Disease / immunology
  • Graft vs Host Disease / pathology
  • Kidney* / drug effects
  • Kidney* / immunology
  • Kidney* / pathology
  • Lupus Erythematosus, Systemic* / drug therapy
  • Lupus Erythematosus, Systemic* / pathology
  • Lymphocyte Activation
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred DBA
  • Oligopeptides / genetics
  • Oligopeptides / pharmacology*
  • Oligopeptides / therapeutic use*
  • T-Lymphocytes / immunology

Substances

  • Autoantibodies
  • Oligopeptides