Roxithromycin downregulates production of CTACK/CCL27 and MIP-3α/CCL20 from epidermal keratinocytes

Arch Dermatol Res. 2010 Dec;302(10):763-7. doi: 10.1007/s00403-010-1068-x. Epub 2010 Jul 13.

Abstract

Cutaneous T cell-attracting chemokine (CTACK)/CCL27 and macrophage inflammatory protein (MIP)-3α/CCL20 are the major inflammatory chemokines involved in skin inflammation. The present study showed that roxithromycin (RXM) suppressed the TNFα-induced production of CCL27 and CCL20 in HaCaT keratinocytes and normal human keratinocytes (NHKs) in a dose-dependent manner. The production of CCL20 induced by TNFα was suppressed by the addition of inhibitors of nuclear factor kappa B (NFκB). RXM suppressed NFκB activity induced by TNFα. RXM, by regulating CCL27 and CCL20, may contribute to the modulation of inflammation.

MeSH terms

  • Cell Line
  • Chemokine CCL20 / genetics
  • Chemokine CCL20 / immunology
  • Chemokine CCL20 / metabolism*
  • Chemokine CCL27 / genetics
  • Chemokine CCL27 / immunology
  • Chemokine CCL27 / metabolism*
  • Dose-Response Relationship, Drug
  • Down-Regulation
  • Epidermis / pathology
  • Humans
  • Immunosuppression Therapy
  • Inflammation
  • Keratinocytes / drug effects*
  • Keratinocytes / immunology
  • Keratinocytes / metabolism
  • Keratinocytes / pathology
  • NF-kappa B / antagonists & inhibitors*
  • Roxithromycin / pharmacology*
  • Tumor Necrosis Factor-alpha / immunology
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Chemokine CCL20
  • Chemokine CCL27
  • NF-kappa B
  • Tumor Necrosis Factor-alpha
  • Roxithromycin