Hyaluronan synthesis mediates the fibrotic response of keratocytes to transforming growth factor beta

J Biol Chem. 2010 Oct 15;285(42):32012-9. doi: 10.1074/jbc.M110.127183. Epub 2010 Aug 4.

Abstract

TGFβ induces fibrosis in healing corneal wounds, and in vitro corneal keratocytes up-regulate expression of several fibrosis-related genes in response to TGFβ. Hyaluronan (HA) accumulates in healing corneas, and HA synthesis is induced by TGFβ by up-regulation of HA synthase 2. This study tested the hypothesis that HA acts as an extracellular messenger, enhancing specific fibrotic responses of keratocytes to TGFβ. HA synthesis inhibitor 4-methylumbelliferone (4MU) blocked TGFβ induction of HA synthesis in a concentration-dependent manner. 4MU also inhibited TGFβ-induced up-regulation of α-smooth muscle actin, collagen type III, and extra domain A-fibronectin. Chemical analogs of 4MU also inhibited fibrogenic responses in proportion to their inhibition of HA synthesis. 4MU, however, showed no effect on TGFβ induction of luciferase by the 3TP-Lux reporter plasmid. Inhibition of HA using siRNA to HA synthase 2 reduced TGFβ up-regulation of smooth muscle actin, fibronectin, and cell division. Similarly, brief treatment of keratocytes with hyaluronidase reduced TGFβ responses. These results suggest that newly synthesized cell-associated HA acts as an extracellular enhancer of wound healing and fibrosis in keratocytes by augmenting a limited subset of the cellular responses to TGFβ.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cattle
  • Cells, Cultured
  • Cornea / cytology
  • Cornea / pathology
  • Fibrosis*
  • Glucuronosyltransferase / genetics
  • Glucuronosyltransferase / metabolism
  • Humans
  • Hyaluronan Synthases
  • Hyaluronic Acid / biosynthesis*
  • Hyaluronoglucosaminidase / metabolism
  • Isoenzymes / genetics
  • Isoenzymes / metabolism
  • Keratinocytes / drug effects*
  • Keratinocytes / pathology*
  • Keratinocytes / physiology
  • Platelet-Derived Growth Factor / pharmacology
  • Signal Transduction / physiology
  • Transforming Growth Factor beta / pharmacology*

Substances

  • Isoenzymes
  • Platelet-Derived Growth Factor
  • Transforming Growth Factor beta
  • Hyaluronic Acid
  • Glucuronosyltransferase
  • Hyaluronan Synthases
  • Hyaluronoglucosaminidase