Small RNAs control sodium channel expression, nociceptor excitability, and pain thresholds

J Neurosci. 2010 Aug 11;30(32):10860-71. doi: 10.1523/JNEUROSCI.1980-10.2010.

Abstract

To examine the role of small RNAs in peripheral pain pathways, we deleted the enzyme Dicer in mouse postmitotic damage-sensing neurons. We used a Nav1.8-Cre mouse to target those nociceptors important for inflammatory pain. The conditional null mice were healthy with a normal number of sensory neurons and normal acute pain thresholds. Behavioral studies showed that inflammatory pain was attenuated or abolished. Inflammatory mediators failed to enhance excitability of Nav1.8+ sensory neurons from null mutant mice. Acute noxious input into the dorsal horn of the spinal cord was apparently normal, but the increased input associated with inflammatory pain measured using c-Fos staining was diminished. Microarray and quantitative real-time reverse-transcription PCR (qRT-PCR) analysis showed that Dicer deletion lead to the upregulation of many broadly expressed mRNA transcripts in dorsal root ganglia. By contrast, nociceptor-associated mRNA transcripts (e.g., Nav1.8, P2xr3, and Runx-1) were downregulated, resulting in lower levels of protein and functional expression. qRT-PCR analysis also showed lowered levels of expression of nociceptor-specific pre-mRNA transcripts. MicroRNA microarray and deep sequencing identified known and novel nociceptor microRNAs in mouse Nav1.8+ sensory neurons that may regulate nociceptor gene expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analysis of Variance
  • Animals
  • Cerebellum / cytology
  • Core Binding Factor Alpha 2 Subunit / genetics
  • Core Binding Factor Alpha 2 Subunit / metabolism
  • DEAD-box RNA Helicases / deficiency
  • Disease Models, Animal
  • Endoribonucleases / deficiency
  • Female
  • Freund's Adjuvant / adverse effects
  • Ganglia, Spinal / metabolism
  • Gene Expression Profiling / methods
  • Gene Expression Regulation / genetics*
  • Male
  • Mice
  • Mice, Knockout
  • MicroRNAs / physiology
  • NAV1.8 Voltage-Gated Sodium Channel
  • Nerve Tissue Proteins / metabolism
  • Nociceptors / metabolism*
  • Oligonucleotide Array Sequence Analysis / methods
  • Pain / chemically induced
  • Pain / genetics
  • Pain / physiopathology*
  • Pain Measurement
  • Pain Threshold / physiology*
  • Proto-Oncogene Proteins c-fos / metabolism
  • Receptors, Purinergic P2 / genetics
  • Receptors, Purinergic P2 / metabolism
  • Receptors, Purinergic P2X3
  • Ribonuclease III
  • Sensory Receptor Cells / physiology*
  • Sodium Channels / deficiency
  • Sodium Channels / genetics
  • Sodium Channels / metabolism*
  • Spinal Cord / physiopathology
  • Time Factors

Substances

  • Core Binding Factor Alpha 2 Subunit
  • MicroRNAs
  • NAV1.8 Voltage-Gated Sodium Channel
  • Nerve Tissue Proteins
  • P2rx3 protein, mouse
  • Proto-Oncogene Proteins c-fos
  • Receptors, Purinergic P2
  • Receptors, Purinergic P2X3
  • Runx1 protein, mouse
  • Scn10a protein, mouse
  • Sodium Channels
  • Freund's Adjuvant
  • Endoribonucleases
  • Dicer1 protein, mouse
  • Ribonuclease III
  • DEAD-box RNA Helicases