Corticotropin-releasing factor regulates TLR4 expression in the colon and protects mice from colitis

Gastroenterology. 2010 Dec;139(6):2083-92. doi: 10.1053/j.gastro.2010.08.024. Epub 2010 Aug 20.

Abstract

Background & aims: Defects in the colonic innate immune response have been associated with inflammatory bowel disease (IBD). Corticotropin-releasing hormone (CRH, or corticotropin-releasing factor [CRF]) is a neuropeptide that mediates the stress response in humans, is an immunomodulatory factor with proinflammatory effects, and regulates transcription of Toll-like receptors (TLR)-2 and TLR4. We investigated the role of CRF in an innate immunity-dependent mouse model of IBD.

Methods: Crh(-/-) and wild-type (Crh(+/+)) mice, which are glucocorticoid insufficient, were given dextran sodium sulfate in their drinking water to induce colitis; in some experiments, mice were also given glucocorticoids. Phenotypes of mice were compared; tissues were analyzed by histology and for expression of immune mediators.

Results: Crh(-/-) mice had more colonic inflammation than Crh(+/+) mice, characterized by reduced numbers of crypts and severe epithelial damage and ulcerations. Colonic tissue levels of the proinflammatory factors interleukin-12 and prostaglandin E(2) were increased in the Crh(-/-) mice. Colons of Crh(-/-) mice expressed lower levels of Tlr4 than wild-type mice before, but not after, colitis was induced. Administration of glucocorticoid at low levels did not prevent Crh(-/-) mice from developing severe colitis. Crh(-/-) mice were unable to recover from acute colitis, as indicated by their increased death rate.

Conclusions: Mice deficient in CRF down-regulate TLR4 and are more susceptible to dextran sodium sulfate-induced colitis. CRF has anti-inflammatory effects in innate immunity-dependent colitis and its recovery phase; these are independent of glucocorticoid administration. CRF might therefore be developed as a therapeutic target for patients with IBD.

MeSH terms

  • Acute Disease
  • Animals
  • Colitis / chemically induced
  • Colitis / immunology*
  • Colitis / mortality
  • Colon / immunology*
  • Corticotropin-Releasing Hormone* / genetics
  • Corticotropin-Releasing Hormone* / immunology
  • Corticotropin-Releasing Hormone* / metabolism
  • Dextran Sulfate / toxicity
  • Disease Models, Animal
  • Kaplan-Meier Estimate
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Mutant Strains
  • Morbidity
  • Stress, Physiological / immunology
  • Toll-Like Receptor 4* / genetics
  • Toll-Like Receptor 4* / immunology
  • Toll-Like Receptor 4* / metabolism

Substances

  • Tlr4 protein, mouse
  • Toll-Like Receptor 4
  • Corticotropin-Releasing Hormone
  • Dextran Sulfate