Efficacy and safety of maraviroc versus efavirenz, both with zidovudine/lamivudine: 96-week results from the MERIT study

HIV Clin Trials. 2010 May-Jun;11(3):125-32. doi: 10.1310/hct1103-125.

Abstract

Background: The MERIT study evaluated maraviroc versus efavirenz, both with zidovudine/lamivudine, in treatment-naïve patients with CCR5-tropic (R5) HIV-1. Post hoc analyses previously assessed week 48 outcomes in patients rescreened with R5 virus by a more sensitive tropism assay.

Methods: Week 96 efficacy (post hoc, n = 614) and safety (n = 721) were assessed.

Results: Proportions of subjects <50 copies/mL (58.8% maraviroc, 62.7% efavirenz) and time to loss of virologic response (TLOVR) responders (<50 copies/mL: 60.5% vs 60.7%) were similar. Maraviroc recipients had greater CD4 increases (+ 212 vs + 171 cells/mm(3)) and fewer adverse event discontinuations (6.1% vs 15.5%), malignancies, and category C events.

Conclusion: Week 96 data confirm week 48 observations in MERIT.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Alkynes
  • Anti-HIV Agents / adverse effects
  • Anti-HIV Agents / therapeutic use*
  • Benzoxazines / adverse effects
  • Benzoxazines / therapeutic use*
  • CCR5 Receptor Antagonists
  • Cyclohexanes / adverse effects
  • Cyclohexanes / therapeutic use*
  • Cyclopropanes
  • Drug Therapy, Combination
  • Female
  • HIV Fusion Inhibitors / adverse effects
  • HIV Fusion Inhibitors / therapeutic use*
  • HIV Infections / drug therapy*
  • HIV Infections / immunology
  • HIV Infections / virology
  • HIV-1*
  • Humans
  • Lamivudine / adverse effects
  • Lamivudine / therapeutic use*
  • Male
  • Maraviroc
  • Middle Aged
  • Treatment Outcome
  • Triazoles / adverse effects
  • Triazoles / therapeutic use*
  • Zidovudine / adverse effects
  • Zidovudine / therapeutic use*

Substances

  • Alkynes
  • Anti-HIV Agents
  • Benzoxazines
  • CCR5 Receptor Antagonists
  • Cyclohexanes
  • Cyclopropanes
  • HIV Fusion Inhibitors
  • Triazoles
  • Lamivudine
  • Zidovudine
  • efavirenz
  • Maraviroc