Small-molecule regulators that mimic transcription factors

Biochim Biophys Acta. 2010 Oct-Dec;1799(10-12):768-74. doi: 10.1016/j.bbagrm.2010.08.010. Epub 2010 Sep 6.

Abstract

Transcription factors (TFs) are responsible for decoding and expressing the information stored in the genome, which dictates cellular function. Creating artificial transcription factors (ATFs) that mimic endogenous TFs is a major goal at the interface of biology, chemistry, and molecular medicine. Such molecular tools will be essential for deciphering and manipulating transcriptional networks that lead to particular cellular states. In this minireview, the framework for the design of functional ATFs is presented and current challenges in the successful implementation of ATFs are discussed.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Review

MeSH terms

  • Animals
  • Humans
  • Peptidomimetics / chemistry*
  • Peptidomimetics / metabolism*
  • Peptidomimetics / pharmacology*
  • Transcription Factors*
  • Transcription, Genetic / drug effects

Substances

  • Peptidomimetics
  • Transcription Factors