Caspase-8 as a therapeutic target in cancer

Cancer Lett. 2013 May 28;332(2):133-40. doi: 10.1016/j.canlet.2010.07.022. Epub 2010 Sep 3.

Abstract

Caspase-8 is an apical caspase which initiates programmed cell death following death receptor ligation. This central role in apoptosis has prompted significant clinical interest in regulating caspase-8 expression and proteolytic activity. However, caspase-8 has also been found to play a number of non-apoptotic roles in cells, such as promoting activation NF-κB signaling, regulating autophagy and altering endosomal trafficking, and enhancing cellular adhesion and migration. Therefore, depending upon the specific cellular context, caspase-8 may either potentiate or suppress tumor malignancy. Accordingly, a marked heterogeneity exists in the expression patterns of caspase-8 among different tumor types. Therapeutics have been developed which can increase caspase-8 expression, yet it remains unclear whether this approach will be beneficial in all cases. Care is warranted, and the role of caspase-8 should be addressed on a case by case basis.

Publication types

  • Review

MeSH terms

  • Apoptosis*
  • Caspase 8 / metabolism*
  • Cell Adhesion
  • Cell Movement
  • Endosomes / metabolism
  • Gene Expression Regulation, Neoplastic*
  • Humans
  • NF-kappa B / metabolism
  • Neoplasm Metastasis
  • Neoplasms / drug therapy*
  • Neoplasms / pathology*

Substances

  • NF-kappa B
  • CASP8 protein, human
  • Caspase 8