CBP/p300 double null cells reveal effect of coactivator level and diversity on CREB transactivation

EMBO J. 2010 Nov 3;29(21):3660-72. doi: 10.1038/emboj.2010.235. Epub 2010 Sep 21.

Abstract

It remains uncertain how the DNA sequence of mammalian genes influences the transcriptional response to extracellular signals. Here, we show that the number of CREB-binding sites (CREs) affects whether the related histone acetyltransferases (HATs) CREB-binding protein (CBP) and p300 are required for endogenous gene transcription. Fibroblasts with both CBP and p300 knocked-out had strongly attenuated histone H4 acetylation at CREB-target genes in response to cyclic-AMP, yet transcription was not uniformly inhibited. Interestingly, dependence on CBP/p300 was often different between reporter plasmids and endogenous genes. Transcription in the absence of CBP/p300 correlated with endogenous genes having more CREs, more bound CREB, and more CRTC2 (a non-HAT coactivator of CREB). Indeed, CRTC2 rescued cAMP-inducible expression for certain genes in CBP/p300 null cells and contributed to the CBP/p300-independent expression of other targets. Thus, endogenous genes with a greater local concentration and diversity of coactivators tend to have more resilient-inducible expression. This model suggests how gene expression patterns could be tuned by altering coactivator availability rather than by changing signal input or transcription factor levels.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation
  • Animals
  • Binding Sites
  • Biomarkers / metabolism
  • Blotting, Western
  • CREB-Binding Protein / physiology*
  • Cells, Cultured
  • Chromatin Immunoprecipitation
  • Cyclic AMP / pharmacology
  • E1A-Associated p300 Protein / physiology*
  • Embryo, Mammalian / cytology
  • Embryo, Mammalian / metabolism
  • Fibroblasts / cytology
  • Fibroblasts / metabolism
  • Gene Expression Profiling
  • Histone Acetyltransferases / metabolism*
  • Histones / metabolism
  • Integrases / metabolism
  • Mice
  • Mice, Knockout
  • Oligonucleotide Array Sequence Analysis
  • Promoter Regions, Genetic / genetics
  • RNA, Messenger / genetics
  • RNA, Small Interfering / pharmacology
  • Reverse Transcriptase Polymerase Chain Reaction
  • Signal Transduction
  • Trans-Activators / antagonists & inhibitors
  • Trans-Activators / genetics
  • Trans-Activators / metabolism*
  • Transcription Factors
  • Transcription, Genetic*

Substances

  • Biomarkers
  • Crtc2 protein, mouse
  • Histones
  • RNA, Messenger
  • RNA, Small Interfering
  • Trans-Activators
  • Transcription Factors
  • Cyclic AMP
  • CREB-Binding Protein
  • E1A-Associated p300 Protein
  • Ep300 protein, mouse
  • Histone Acetyltransferases
  • Cre recombinase
  • Integrases