RNA-binding protein HuR regulates RGS4 mRNA stability in rabbit colonic smooth muscle cells

Am J Physiol Cell Physiol. 2010 Dec;299(6):C1418-29. doi: 10.1152/ajpcell.00093.2010. Epub 2010 Sep 29.

Abstract

Regulator of G protein signaling 4 (RGS4) regulates the strength and duration of G protein signaling and plays an important role in smooth muscle contraction, cardiac development, and psychiatric disorders. Little is known about the posttranscriptional regulation of RGS4 expression. We cloned the full-length cDNA of rabbit RGS4, which contains a long 3'-untranslated region (UTR) with several AU-rich elements (AREs). We determined whether RGS4 mRNA stability is mediated by the RNA-binding protein human antigen R (HuR) and contributes to IL-1β-induced upregulation of RGS4 expression. We show that IL-1β treatment in colonic smooth muscle cells doubled the half-life of RGS4 mRNA. Addition of RGS4 3'-UTR to the downstream of Renilla luciferase reporter induced dramatic reduction in the enzyme activity and mRNA expression of luciferase, which was attenuated by the site-directed mutation of the two 3'-most ARE sites. IL-1β increased luciferase mRNA stability in a UTR-dependent manner. Knockdown of HuR significantly aggravated UTR-mediated instability of luciferase and inhibited IL-1β-induced upregulation of RGS4 mRNA. In addition, IL-1β increased cytosolic translocation and RGS4 mRNA binding of HuR. These findings suggest that 3'-most ARE sites within RGS4 3'-UTR are essential for the instability of RGS4 mRNA and IL-1β promotes the stability of RGS4 mRNA through HuR.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • 3' Untranslated Regions
  • Animals
  • Antigens, Surface / genetics
  • Antigens, Surface / metabolism*
  • Base Sequence
  • Colon / metabolism*
  • ELAV Proteins
  • ELAV-Like Protein 1
  • Humans
  • Interleukin-1beta / metabolism*
  • Interleukin-1beta / pharmacology
  • Molecular Sequence Data
  • Myocytes, Smooth Muscle / metabolism*
  • RGS Proteins / genetics
  • RGS Proteins / metabolism*
  • RNA Stability*
  • RNA-Binding Proteins / genetics
  • RNA-Binding Proteins / metabolism*
  • Rabbits
  • Up-Regulation

Substances

  • 3' Untranslated Regions
  • Antigens, Surface
  • ELAV Proteins
  • ELAV-Like Protein 1
  • ELAVL1 protein, human
  • Interleukin-1beta
  • RGS Proteins
  • RNA-Binding Proteins
  • RGS4 protein