Syk is a dual-specificity kinase that self-regulates the signal output from the B-cell antigen receptor

Proc Natl Acad Sci U S A. 2010 Oct 26;107(43):18563-8. doi: 10.1073/pnas.1009048107. Epub 2010 Oct 12.

Abstract

Upon B-cell activation, the signaling subunits Ig-α and Ig-β of the B-cell antigen receptor become phosphorylated not only on tyrosines but also on serine residues. Using a specific antibody, we show that serine 197 (S197) in the cytoplasmic tail of Ig-α is phosphorylated upon B-cell antigen receptor activation, and that this modification inhibits the signal output of the B-cell antigen receptor. Surprisingly, we found that the well-known protein tyrosine kinase Syk (spleen tyrosine kinase) phosphorylates S197 on Ig-α, thus not only activating but also inhibiting signaling from the B-cell antigen receptor. This finding identifies Syk as a dual-specificity kinase and establishes a previously unexplored paradigm for the self-regulation of biological signaling processes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • B-Lymphocytes / immunology*
  • B-Lymphocytes / metabolism*
  • CD79 Antigens / chemistry
  • CD79 Antigens / genetics
  • CD79 Antigens / metabolism
  • Cell Line
  • Drosophila
  • Intracellular Signaling Peptides and Proteins / chemistry
  • Intracellular Signaling Peptides and Proteins / genetics
  • Intracellular Signaling Peptides and Proteins / metabolism*
  • Mice
  • Mice, Inbred BALB C
  • Mice, Knockout
  • Mice, Transgenic
  • Models, Molecular
  • Molecular Sequence Data
  • Mutation
  • Phosphorylation
  • Protein-Tyrosine Kinases / chemistry
  • Protein-Tyrosine Kinases / genetics
  • Protein-Tyrosine Kinases / metabolism*
  • Receptors, Antigen, B-Cell / chemistry
  • Receptors, Antigen, B-Cell / genetics
  • Receptors, Antigen, B-Cell / metabolism*
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism
  • Serine / chemistry
  • Signal Transduction
  • Structural Homology, Protein
  • Syk Kinase

Substances

  • CD79 Antigens
  • Cd79a protein, mouse
  • Intracellular Signaling Peptides and Proteins
  • Receptors, Antigen, B-Cell
  • Recombinant Proteins
  • Serine
  • Protein-Tyrosine Kinases
  • Syk Kinase
  • Syk protein, mouse