The glucagon-like peptide 1 receptor agonist exendin-4 improves reference memory performance and decreases immobility in the forced swim test

Eur J Pharmacol. 2011 Jan 10;650(1):249-55. doi: 10.1016/j.ejphar.2010.10.008. Epub 2010 Oct 14.

Abstract

We have earlier shown that the glucagon-like peptide 1 receptor agonist exendin-4 stimulates neurogenesis in the subventricular zone and excerts anti-parkinsonian behavior. The aim of this study was to assess the effects of exendin-4 treatment on hippocampus-associated cognitive and mood-related behavior in adult rodents. To investigate potential effects of exendin-4 on hippocampal function, radial maze and forced swim test were employed. The time necessary to solve a radial maze task and the duration of immobility in the forced swim test were significantly reduced compared to respective vehicle groups if the animals had received exendin-4 during 1-2weeks before testing. In contrast to the positive control imipramine, single administration of exendin-4 1h before the challenge in the forced swim test had no effect. Immunohistochemical analysis showed that the incorporation of bromodeoxyuridine, a marker for DNA synthesis, as well as doublecortin expression was increased in the hippocampal dentate gyrus following chronic treatment with exendin-4 compared to vehicle-treated controls. The neurogenic effect of exendin-4 on hippocampus was confirmed by quantitative PCR showing an upregulation of mRNA expression for Ki-67, doublecortin and Mash-1. Since exendin-4 significantly improves hippocampus-associated behavior in adult rodents, it may be a candidate for alleviation of mood and cognitive disorders.

MeSH terms

  • Affect / drug effects
  • Affect / physiology
  • Animals
  • Behavior, Animal / drug effects*
  • Behavior, Animal / physiology*
  • Biomarkers / metabolism
  • Bromodeoxyuridine / pharmacology
  • Cell Differentiation / drug effects
  • Cognition / drug effects
  • Cognition / physiology
  • Dose-Response Relationship, Drug
  • Doublecortin Protein
  • Drug Synergism
  • Exenatide
  • Glucagon-Like Peptide-1 Receptor
  • Hippocampus / drug effects
  • Hippocampus / physiology
  • Male
  • Maze Learning / drug effects
  • Maze Learning / physiology
  • Memory / drug effects*
  • Memory / physiology*
  • Neurons / cytology
  • Neurons / drug effects
  • Peptides / pharmacology*
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Glucagon / agonists*
  • Swimming*
  • Venoms / pharmacology*

Substances

  • Biomarkers
  • Dcx protein, rat
  • Doublecortin Protein
  • Glp1r protein, rat
  • Glucagon-Like Peptide-1 Receptor
  • Peptides
  • Receptors, Glucagon
  • Venoms
  • Exenatide
  • Bromodeoxyuridine