Effectiveness of sulfur-containing antioxidants in delaying skeletal muscle fatigue

Med Sci Sports Exerc. 2011 Jun;43(6):1025-31. doi: 10.1249/MSS.0b013e3182019a78.

Abstract

Reactions involving thiol biochemistry seem to play a crucial role in skeletal muscle fatigue. N-acetylcysteine amide (NACA) and L-ergothioneine (ERGO) are thiol-based antioxidants available for human use that have not been evaluated for effects on muscle fatigue.

Purpose: To test the hypothesis that NACA and ERGO delay skeletal muscle fatigue.

Methods: We exposed mouse diaphragm fiber bundles to buffer (CTRL), NACA, ERGO, or N-acetylcysteine (NAC; positive control). Treatments were performed in vitro using 10 mM for 60 min at 37 °C. After treatment, we determined the muscle force-frequency and fatigue characteristics.

Results: The force-frequency relationship was shifted to the left by ERGO and to the right by NACA compared with CTRL and NAC. Maximal tetanic force was similar among groups. The total force-time integral (FTI; N · s · cm) during the fatigue trial was decreased by NACA (420 ± 35, P < 0.05), unaffected by ERGO (657 ± 53), and increased by NAC (P < 0.05) compared with CTRL (581 ± 54). The rate of contraction (dF/dtMAX) during the fatigue trial was not affected by any of the treatments tested. NAC, but not NACA or ERGO, delayed the slowing of muscle relaxation (dF/dtMIN) during fatigue.

Conclusions: In summary, NACA and ERGO did not delay skeletal muscle fatigue in vitro. We conclude that these antioxidants are unlikely to improve human exercise performance.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Acetylcysteine / analogs & derivatives*
  • Acetylcysteine / pharmacology
  • Animals
  • Antioxidants / pharmacology*
  • Diaphragm / drug effects*
  • Ergothioneine / pharmacology*
  • Mice
  • Mice, Inbred C57BL
  • Muscle Fatigue / drug effects*
  • Muscle Relaxation / drug effects

Substances

  • Antioxidants
  • N-Acetylcysteinamide
  • Ergothioneine
  • Acetylcysteine