[Protective activity of Ingavirin in experimental lethal influenza due to pandemic influenza virus A (H1N1)v in albino mice]

Antibiot Khimioter. 2010;55(5-6):24-31.
[Article in Russian]

Abstract

Despite obvious success in the vaccine development and chemotherapy of influenza, it remains a poorly controlled infection leading to emergence of new pandemic variants of the virus with high morbidity and mortality. We investigated the protective activity of Ingavirin against the lethal influenza A (H1N1) 2009 virus infection on albino mice. Oral use of Ingavirin resulted in sharp decreasing of the mortality (index of protection up to 57%), slight decreasing of the infectious titer of the virus in the lungs (up to 40-fold), normalizing of the body weight dynamics and the lung tissue structure vs. the placebo-treated control. The degree of the bronchial epithelium damage was also strongly decreased. The results allow to consider Ingavirin as an effective antiviral against the current pandemic influenza virus.

MeSH terms

  • Amides / therapeutic use*
  • Animals
  • Antiviral Agents / therapeutic use*
  • Caproates
  • Dicarboxylic Acids / therapeutic use*
  • Female
  • Imidazoles / therapeutic use*
  • Influenza A Virus, H1N1 Subtype / drug effects*
  • Influenza A Virus, H1N1 Subtype / physiology
  • Lung / drug effects
  • Lung / pathology
  • Lung / virology
  • Mice
  • Orthomyxoviridae Infections / drug therapy*
  • Orthomyxoviridae Infections / mortality
  • Orthomyxoviridae Infections / virology
  • Virus Replication / drug effects

Substances

  • Amides
  • Antiviral Agents
  • Caproates
  • Dicarboxylic Acids
  • Imidazoles
  • pentanedioic acid imidazolyl ethanamide