Synthesis and antifungal activity of some substituted phenothiazines and related compounds

Eur J Med Chem. 2011 Jan;46(1):101-5. doi: 10.1016/j.ejmech.2010.10.019. Epub 2010 Oct 27.

Abstract

Several phenothiazines and related compounds were synthesized and their antifungal activity was evaluated in vitro. The results observed for α-chloro-N-acetyl phenothiazine led us to choose this compound as a lead in the search of antifungal agents.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antifungal Agents / chemical synthesis*
  • Antifungal Agents / chemistry
  • Antifungal Agents / pharmacology*
  • Drug Discovery
  • Fungi / drug effects
  • Microbial Sensitivity Tests
  • Phenothiazines / chemical synthesis*
  • Phenothiazines / chemistry
  • Phenothiazines / pharmacology*
  • Structure-Activity Relationship

Substances

  • Antifungal Agents
  • Phenothiazines
  • phenothiazine