Advances in microbicide vaginal rings

Antiviral Res. 2010 Dec:88 Suppl 1:S30-9. doi: 10.1016/j.antiviral.2010.09.003.

Abstract

Vaginal ring devices capable of providing sustained/controlled release of incorporated actives are already marketed for steroidal contraception and estrogen replacement therapy. In recent years, there has been considerable interest in developing similar ring devices for the administration of microbicidal compounds to prevent vaginal HIV transmission. Intended to be worn continuously, such coitally independent microbicide rings are being developed to maintain effective vaginal microbicide concentrations over many weeks or months, thereby overcoming issues around timing of product application, user compliance and acceptability associated with more conventional semi-solid formulations. In this article, an overview of vaginal ring technologies is presented, followed by a review of recent advances and issues pertaining to their application for the delivery of HIV microbicides. This article forms part of a special supplement on presentations covering intravaginal rings, based on the symposium "Trends in Microbicide Formulations", held on 25 and 26 January 2010, Arlington, VA.

Publication types

  • Review

MeSH terms

  • Administration, Intravaginal
  • Anti-HIV Agents / administration & dosage*
  • Anti-HIV Agents / chemistry
  • Anti-HIV Agents / therapeutic use
  • Anti-Infective Agents / administration & dosage*
  • Anti-Infective Agents / chemistry
  • Anti-Infective Agents / therapeutic use
  • Chemistry, Pharmaceutical
  • Coated Materials, Biocompatible / chemistry*
  • Coated Materials, Biocompatible / standards
  • Coated Materials, Biocompatible / therapeutic use*
  • Contraceptive Devices, Female / economics*
  • Contraceptive Devices, Female / standards*
  • Contraceptive Devices, Female / virology*
  • Costs and Cost Analysis
  • Dosage Forms
  • Drug and Narcotic Control
  • Female
  • HIV / drug effects*
  • HIV Infections / drug therapy
  • HIV Infections / prevention & control*
  • HIV Infections / transmission
  • Humans
  • Male
  • Risk Factors
  • Vagina / drug effects
  • Vagina / virology

Substances

  • Anti-HIV Agents
  • Anti-Infective Agents
  • Coated Materials, Biocompatible
  • Dosage Forms