Real time, high resolution video imaging of apoptosis in single cells with a polymeric nanoprobe

Bioconjug Chem. 2011 Feb 16;22(2):125-31. doi: 10.1021/bc1004119. Epub 2011 Jan 10.

Abstract

We report a new apoptosis nanoprobe (Apo-NP) designed on the basis of a polymer nanoparticle platform. This simple one-step technique is capable of boosting fluorescence signals upon apoptosis in living cells, enabling real-time imaging of apoptosis in single cells and in vivo. The Apo-NP efficiently delivers chemically labeled, dual-quenched caspase-3-sensitive fluorogenic peptides into cells, allowing caspase-3-dependent strong fluorescence amplification to be imaged in apoptotic cells in real-time and at high resolution. The design platform of the Apo-NP is flexible and can be fine-tuned for a wide array of applications such as identification of caspase-related apoptosis in pathologies and for monitoring therapeutic efficacy of apoptotic drugs in cancer treatment.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology
  • Apoptosis* / drug effects
  • Caspase 3 / chemistry
  • Caspase 3 / metabolism
  • Doxorubicin / pharmacology
  • Fluorescent Dyes / administration & dosage
  • Fluorescent Dyes / chemistry*
  • Humans
  • Luminescent Measurements
  • Mice
  • Molecular Imaging*
  • Molecular Structure
  • Nanoparticles / administration & dosage
  • Nanoparticles / chemistry*
  • Neoplasms, Experimental
  • Particle Size
  • Polymers / administration & dosage
  • Polymers / chemistry*
  • Surface Properties
  • Tumor Cells, Cultured

Substances

  • Antineoplastic Agents
  • Fluorescent Dyes
  • Polymers
  • Doxorubicin
  • Caspase 3