Phosphorylation of glutamyl-prolyl tRNA synthetase by cyclin-dependent kinase 5 dictates transcript-selective translational control

Proc Natl Acad Sci U S A. 2011 Jan 25;108(4):1415-20. doi: 10.1073/pnas.1011275108. Epub 2011 Jan 10.

Abstract

Cyclin-dependent kinase 5 (Cdk5) is an atypical but essential member of the Cdk kinase family, and its dysregulation or deletion has been implicated in inflammation-related disorders by an undefined mechanism. Here we show that Cdk5 is an indispensable activator of the GAIT (IFN-γ-activated inhibitor of translation) pathway, which suppresses expression of a posttranscriptional regulon of proinflammatory genes in myeloid cells. Through induction of its regulatory protein, Cdk5R1 (p35), IFN-γ activates Cdk5 to phosphorylate Ser(886) in the linker domain of glutamyl-prolyl tRNA synthetase (EPRS), the initial event in assembly of the GAIT complex. Cdk5/p35 also induces, albeit indirectly via a distinct kinase, phosphorylation of Ser(999), the second essential event in GAIT pathway activation. Diphosphorylated EPRS is released from its residence in the tRNA multisynthetase complex for immediate binding to NS1-associated protein and subsequent binding to ribosomal protein L13a and GAPDH. The mature heterotetrameric GAIT complex binds the 3' UTR GAIT element of VEGF-A and other target mRNAs and suppresses their translation in myeloid cells. Inhibition of Cdk5/p35 inhibits both EPRS phosphorylation events, prevents EPRS release from the tRNA multisynthetase complex, and blocks translational suppression of GAIT element-bearing mRNAs, resulting in increased expression of inflammatory proteins. Our study reveals a unique role of Cdk5/p35 in activation of the major noncanonical function of EPRS, namely translational control of macrophage inflammatory gene expression.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acyl-tRNA Synthetases / genetics
  • Amino Acyl-tRNA Synthetases / metabolism*
  • Cyclin-Dependent Kinase 5 / genetics
  • Cyclin-Dependent Kinase 5 / metabolism
  • Humans
  • Immunoblotting
  • Interferon-gamma / pharmacology
  • Nerve Tissue Proteins / genetics
  • Nerve Tissue Proteins / metabolism
  • Phosphorylation / drug effects
  • Protein Binding
  • Protein Biosynthesis / drug effects
  • Protein Biosynthesis / genetics*
  • RNA Interference
  • Reverse Transcriptase Polymerase Chain Reaction
  • Ribosomal Proteins / metabolism
  • Serine / genetics
  • Serine / metabolism*
  • Transcription, Genetic / drug effects
  • Transcription, Genetic / genetics*
  • U937 Cells
  • Vascular Endothelial Growth Factor A / genetics
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • Nerve Tissue Proteins
  • Ribosomal Proteins
  • Vascular Endothelial Growth Factor A
  • neuronal Cdk5 activator (p25-p35)
  • Serine
  • Interferon-gamma
  • Cyclin-Dependent Kinase 5
  • Amino Acyl-tRNA Synthetases
  • glutamyl-prolyl-tRNA synthetase