The cation channel mucolipin-1 is a bifunctional protein that facilitates membrane remodeling via its serine lipase domain

Exp Cell Res. 2011 Apr 1;317(6):691-705. doi: 10.1016/j.yexcr.2011.01.008. Epub 2011 Jan 20.

Abstract

Phospholipase modulators have been shown to affect the topology of lipid bilayers and the formation of tubulo-vesicular structures, but the specific endogenous phospholipases involved have yet to be identified. Here we show that TRPML1 (MLN1), a Ca(2+)-permeable channel, contributes to membrane remodeling through a serine lipase consensus domain, and thus represents a novel type of bifunctional protein. Remarkably, this serine lipase active site determines the ability of MLN1 to generate tubulo-vesicular extensions in mucolipin-1-expressing oocytes, human fibroblasts and model membrane vesicles. Our demonstration that MLN1 is involved in membrane remodeling and the formation of extensions suggests that it may play a role in the formation of cellular processes linked to the late endosome/lysosome (LE/L) pathway. MLN1 is absent or mutated in patients with mucolipidosis IV (MLIV), a lysosomal disorder with devastating neurological and other consequences. This study provides potential insight into the pathophysiology of MLIV.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Membrane / chemistry*
  • Cell Membrane / metabolism*
  • Fibroblasts / chemistry
  • Fibroblasts / enzymology
  • Fibroblasts / metabolism
  • Humans
  • Lipase / genetics
  • Lipase / metabolism*
  • Membrane Fusion Proteins / genetics
  • Membrane Fusion Proteins / metabolism
  • Mucolipidoses / enzymology
  • Mutation
  • Protein Structure, Tertiary
  • TRPM Cation Channels / genetics
  • TRPM Cation Channels / metabolism*
  • Transient Receptor Potential Channels
  • Xenopus laevis

Substances

  • MCOLN1 protein, human
  • Membrane Fusion Proteins
  • TRPM Cation Channels
  • Transient Receptor Potential Channels
  • Lipase