Histone deacetylase (HDAC) inhibition as a novel treatment for diabetes mellitus

Mol Med. 2011 May-Jun;17(5-6):378-90. doi: 10.2119/molmed.2011.00021. Epub 2011 Jan 25.

Abstract

Both common forms of diabetes have an inflammatory pathogenesis in which immune and metabolic factors converge on interleukin-1β as a key mediator of insulin resistance and β-cell failure. In addition to improving insulin resistance and preventing β-cell inflammatory damage, there is evidence of genetic association between diabetes and histone deacetylases (HDACs); and HDAC inhibitors (HDACi) promote β-cell development, proliferation, differentiation and function and positively affect late diabetic microvascular complications. Here we review this evidence and propose that there is a strong rationale for preclinical studies and clinical trials with the aim of testing the utility of HDACi as a novel therapy for diabetes.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / therapeutic use
  • Diabetes Mellitus / drug therapy
  • Diabetes Mellitus / enzymology*
  • Diabetes Mellitus / metabolism*
  • Histone Deacetylase Inhibitors / therapeutic use
  • Histone Deacetylases / genetics
  • Histone Deacetylases / metabolism*
  • Humans
  • Interleukin-1beta / metabolism

Substances

  • Anti-Inflammatory Agents
  • Histone Deacetylase Inhibitors
  • Interleukin-1beta
  • Histone Deacetylases