Effect of ethinylestradiol/cyproterone acetate on endothelial function in young non-obese women with polycystic ovary syndrome: a pilot study

Gynecol Endocrinol. 2011 Sep;27(9):615-21. doi: 10.3109/09513590.2010.521265. Epub 2011 Feb 17.

Abstract

Background: Combined oral contraceptives are used in polycystic ovary syndrome (PCOS) women for the treatment of hyperandrogenism and menstrual cycle disturbances.

Aim: To assess the effect of ethinylestradiol and cyproterone acetate (EE/CA) on endothelial function in young, non-obese PCOS women in a pilot study.

Methods: Thirteen young, non-obese PCOS women (20.9 ± 3.7 years, 23.0 ± 4.0 kg/m(2)) received 35 mcg EE & 2 mg CA for 6 months. Fourteen age- and body mass index (BMI)-matched healthy women served as controls. Endothelial function assessed by brachial artery flow-mediated dilation (FMD), indices of hyperandrogenism, and insulin resistance were studied at baseline and 6-month follow-up.

Results: FMD was impaired in PCOS compared to control women (4.67 ± 2.38% vs. 10.12 ± 3.19%, p < 0.001), but increased significantly following EE/CA (9.99 ± 2.11%, p < 0.001 vs. baseline), reaching normal values (p = NS vs. controls). EE/CA also significantly decreased hyperandrogenism indices and increased total and HDL cholesterol and triglycerides (p < 0.05 vs. baseline). The only independent predictor of treatment-induced FMD improvement in PCOS women was the decrease in free androgen index.

Conclusions: Treatment with combination of estrogens and antiandrogens reverses endothelial dysfunction in young, non-obese PCOS women mainly via improving hyperandrogenism. Further research is needed to investigate whether this treatment may also reduce cardiovascular risk in these women.

Publication types

  • Clinical Trial

MeSH terms

  • Adolescent
  • Adult
  • Androgen Antagonists / pharmacology
  • Androgen Antagonists / therapeutic use*
  • Cyproterone Acetate / pharmacology
  • Cyproterone Acetate / therapeutic use*
  • Drug Therapy, Combination
  • Estrogens / pharmacology
  • Estrogens / therapeutic use*
  • Ethinyl Estradiol / pharmacology
  • Ethinyl Estradiol / therapeutic use*
  • Female
  • Humans
  • Pilot Projects
  • Polycystic Ovary Syndrome / drug therapy*
  • Prospective Studies
  • Regression Analysis
  • Vasodilation / drug effects*
  • Young Adult

Substances

  • Androgen Antagonists
  • Estrogens
  • Ethinyl Estradiol
  • Cyproterone Acetate