Sirolimus prevents short-term renal changes induced by ischemia-reperfusion injury in rats

Am J Nephrol. 2011;33(3):239-49. doi: 10.1159/000324577. Epub 2011 Feb 28.

Abstract

Background: Ischemia-reperfusion (I/R) is present at various degrees in kidney transplants. I/R plays a major role in early function and long-term survival of renal allograft. The purpose of our study was to determine if immunosuppressants modulate I/R in a model that separates I/R from all immune responses.

Methods: Sprague-Dawley rats with monolateral renal I/R received daily cyclosporine (A), tacrolimus (B), sirolimus (C) or saline (D). Sham-operated rats received saline (E). After 30 days, glomerular filtration rate for each kidney was measured by inulin clearance. Kidney injury was examined, and TGF-β, fibronectin and metalloproteases were evaluated by real-time PCR, Western blot and zymography.

Results: Sirolimus, but not cyclosporine and tacrolimus, prevented a glomerular filtration rate decrease in I/R kidneys (403 ± 303 vs. 1,006 ± 484 μl/min, p < 0.05; 126 ± 170 vs. 567 ± 374 μl/min, p < 0.05; 633 ± 293 vs. 786 ± 255; A, B and C group, respectively, I/R vs. contralateral kidneys). Sirolimus reduced ED-1+ cell infiltrate, interstitial fibrosis and intimal thickening of small vessels observed in I/R kidneys of controls and calcineurin inhibitor-treated rats. Tacrolimus and cyclosporine increased fibronectin and TGF-β expression and matrix deposition. Only sirolimus increased metalloprotease activity.

Conclusions: Sirolimus but not calcineurin inhibitors prevented I/R-induced kidney injury.

MeSH terms

  • Animals
  • Cyclosporine / therapeutic use*
  • Glomerular Filtration Rate
  • Immunosuppressive Agents / therapeutic use*
  • Kidney / pathology
  • Kidney Diseases / pathology
  • Kidney Diseases / prevention & control*
  • Kidney Function Tests
  • Male
  • Rats
  • Rats, Sprague-Dawley
  • Reperfusion Injury / pathology
  • Reperfusion Injury / prevention & control*
  • Sirolimus / therapeutic use*
  • Tacrolimus / therapeutic use*

Substances

  • Immunosuppressive Agents
  • Cyclosporine
  • Sirolimus
  • Tacrolimus