Activation of P-TEFb at sites of dual HIV/TB infection, and inhibition of MTB-induced HIV transcriptional activation by the inhibitor of CDK9, Indirubin-3'-monoxime

AIDS Res Hum Retroviruses. 2012 Feb;28(2):182-7. doi: 10.1089/aid.2010.0211. Epub 2011 May 6.

Abstract

At sites of Mycobacterium tuberculosis (MTB) infection, HIV-1 replication is increased during tuberculosis (TB). Here we investigated the role of positive transcription elongation factor (P-TEFb), comprised of CycT1 and CDK9, as the cellular cofactor of HIV-1 Tat protein in transcriptional activation of HIV-1 in mononuclear cells from HIV-1-infected patients with pleural TB. Expression of CycT1 in response to MTB was assessed in mononuclear cells from pleural fluid (PFMC) and blood (PBMC) from HIV/TB patients with pleural TB, and in blood monocytes (MN) from singly infected HIV-1-seropositive subjects. We then examined whether the CDK9 inhibitor, Indirubin 3'-monoxime (IM), was effective in inhibition of MTB-induced HIV-1 mRNA expression. We found higher expression of CycT1 mRNA in PFMCs as compared to PBMCs from HIV/TB-coinfected subjects. MTB induced the expression of CycT1 and HIV-1 gag/pol mRNA in both PFMCs from HIV/TB subjects and MN from HIV-1-infected subjects. CycT1 protein was also induced by MTB stimulation in PFMCs from HIV/TB patients, and both MN and in vitro-derived macrophages. Inhibition of CDK9 by IM in both PFMCs from HIV/TB and MN from HIV-1-infected subjects in response to MTB led to inhibition of HIV-1 mRNA expression. These data imply that IM may be useful as an adjunctive therapy in control of HIV-1 replication in HIV/TB dually infected subjects.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Blotting, Western
  • Coinfection
  • Cyclin T / drug effects
  • Female
  • HIV Infections / drug therapy
  • HIV Infections / genetics
  • HIV Infections / metabolism*
  • HIV-1 / drug effects
  • HIV-1 / physiology*
  • Humans
  • Indoles / pharmacokinetics*
  • Male
  • Middle Aged
  • Mycobacterium tuberculosis / drug effects*
  • Mycobacterium tuberculosis / metabolism
  • Oximes / pharmacokinetics*
  • Positive Transcriptional Elongation Factor B / drug effects
  • Positive Transcriptional Elongation Factor B / genetics
  • Positive Transcriptional Elongation Factor B / metabolism*
  • Transcriptional Activation / drug effects
  • Tuberculosis / drug therapy
  • Tuberculosis / genetics
  • Tuberculosis / metabolism*
  • Uganda / epidemiology
  • Virus Replication / drug effects

Substances

  • Cyclin T
  • Indoles
  • Oximes
  • indirubin-3'-monoxime
  • Positive Transcriptional Elongation Factor B