Suppression of indomethacin-induced apoptosis in the small intestine due to Bach1 deficiency

Free Radic Res. 2011 Jun;45(6):717-27. doi: 10.3109/10715762.2011.574287. Epub 2011 Apr 8.

Abstract

BTB and CNC homologue 1 (Bach1) is a transcriptional repressor of heme oxygenase-1 (HO-1). This study hypothesized that Bach1 plays an important role in the indomethacin-induced apoptosis in the case of small-intestinal mucosal injury. Eight-week-old male C57BL/6 (wild-type) and homozygous Bach1-deficient C57BL/6 mice were included in this study. Mucosal injuries induced by subcutaneously administering indomethacin were evaluated macroscopically, histologically and biochemically. Indomethacin-induced injuries were improved in Bach1-deficient mice. Immunohistochemistry showed an increase in the number of HO-1-positive cells, which were mainly F4/80 positive macrophages, in Bach1-deficient mice. Indomethacin administration increased the expression of HO-1 mRNA and protein in the small intestine in Bach1-deficient mice. Terminal deoxynucleotidyl transferase-mediated dUTP nick end labelling (TUNEL) staining showed that the extent of apoptosis was suppressed in Bach1-deficent mice. In conclusion, deficiency of the Bach1 gene inhibited apoptosis and thus suppressed mucosal injury, indicating that Bach1 is a novel therapeutic target for indomethacin-induced intestinal injury.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects*
  • Basic-Leucine Zipper Transcription Factors / deficiency*
  • Basic-Leucine Zipper Transcription Factors / genetics
  • Caspase 3 / metabolism
  • Enzyme Activation
  • Enzyme Assays
  • Gene Deletion
  • Heme Oxygenase-1 / antagonists & inhibitors
  • Heme Oxygenase-1 / genetics
  • Heme Oxygenase-1 / metabolism
  • Ileum / drug effects*
  • Ileum / metabolism
  • Ileum / pathology
  • Indomethacin / adverse effects*
  • Male
  • Metalloporphyrins / pharmacology
  • Mice
  • Mice, Inbred C57BL
  • Protoporphyrins / pharmacology
  • Tumor Necrosis Factor-alpha / genetics
  • Tumor Necrosis Factor-alpha / metabolism
  • Ulcer / chemically induced
  • Ulcer / pathology*

Substances

  • Bach1 protein, mouse
  • Basic-Leucine Zipper Transcription Factors
  • Metalloporphyrins
  • Protoporphyrins
  • Tumor Necrosis Factor-alpha
  • tin protoporphyrin IX
  • Heme Oxygenase-1
  • Caspase 3
  • Indomethacin