Dearomatization strategies in the synthesis of complex natural products

Angew Chem Int Ed Engl. 2011 Apr 26;50(18):4068-93. doi: 10.1002/anie.201006017. Epub 2011 Apr 19.

Abstract

Evolution in the field of the total synthesis of natural products has led to exciting developments over the last decade. Numerous chemoselective and enantioselective methodologies have emerged from total syntheses, resulting in efficient access to many important natural product targets. This Review highlights recent developments concerning dearomatization, a powerful strategy for the total synthesis of architecturally complex natural products wherein planar, aromatic scaffolds are converted to three-dimensional molecular architectures.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Review

MeSH terms

  • Biological Products / chemical synthesis*
  • Biological Products / chemistry
  • Furans / chemical synthesis
  • Furans / chemistry
  • Indoles / chemical synthesis
  • Indoles / chemistry
  • Phenols / chemistry
  • Pyrroles / chemical synthesis
  • Pyrroles / chemistry
  • Stereoisomerism

Substances

  • Biological Products
  • Furans
  • Indoles
  • Phenols
  • Pyrroles