Effects of lowered serotonin transmission on cocaine-induced striatal dopamine response: PET [¹¹C]raclopride study in humans

Br J Psychiatry. 2011 Nov;199(5):391-7. doi: 10.1192/bjp.bp.110.084178. Epub 2011 May 4.

Abstract

Background: Low serotonin transmission is thought to increase susceptibility to a wide range of substance use disorders and impulsive traits.

Aims: To investigate the effects of lowered serotonin on cocaine-induced (1.0 mg/kg cocaine, self-administered intranasally) dopamine responses and drug craving.

Method: In non-dependent cocaine users, serotonin transmission was reduced using the acute tryptophan depletion method. Striatal dopamine responses were measured using positron emission tomography with [(11)C]raclopride.

Results: Acute tryptophan depletion increased drug craving and striatal dopamine responses to cocaine. These acute tryptophan depletion-induced increases did not occur in the absence of cocaine.

Conclusions: The results suggest that low serotonin transmission can increase dopaminergic and appetitive responses to cocaine. These findings might identify a mechanism by which individuals with low serotonin are at elevated risk for both substance use disorders and comorbid conditions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Intranasal
  • Adult
  • Analysis of Variance
  • Cocaine / administration & dosage
  • Cocaine / metabolism
  • Cocaine / pharmacology*
  • Cocaine-Related Disorders / diagnostic imaging
  • Cocaine-Related Disorders / metabolism*
  • Cocaine-Related Disorders / psychology
  • Corpus Striatum / diagnostic imaging
  • Corpus Striatum / drug effects
  • Corpus Striatum / metabolism*
  • Dopamine / metabolism*
  • Dopamine Uptake Inhibitors / administration & dosage
  • Dopamine Uptake Inhibitors / metabolism
  • Dopamine Uptake Inhibitors / pharmacology*
  • Female
  • Humans
  • Magnetic Resonance Imaging
  • Male
  • Positron-Emission Tomography / methods
  • Raclopride / pharmacokinetics
  • Radiopharmaceuticals / pharmacokinetics
  • Serotonin / metabolism*
  • Tryptophan / administration & dosage
  • Tryptophan / deficiency
  • Tryptophan / metabolism
  • Young Adult

Substances

  • Dopamine Uptake Inhibitors
  • Radiopharmaceuticals
  • Serotonin
  • Raclopride
  • Tryptophan
  • Cocaine
  • Dopamine