Erythroid membrane-bound protein kinase binds to a membrane component and is regulated by phosphatidylinositol 4,5-bisphosphate

J Biol Chem. 1990 May 5;265(13):7369-76.

Abstract

In the erythrocyte, a membrane-bound serine/threonine protein kinase (a casein kinase) has been shown to phosphorylate a number of membrane proteins, modulating their function. Here we report that the membrane-bound protein kinase binds to membranes by an association with a minor membrane component contained in preparations of glycophorin (possibly a minor glycophorin). The binding of the kinase to glycophorins does not significantly modify kinase activity. However, upon binding, the kinase activity is potently inhibited by phosphatidylinositol 4,5-bisphosphate, and the affinity of the kinase for the glycophorins is increased. Other phospholipids or polyanions such as inositol 1,4,5-trisphosphate or 2,3-diphosphoglycerate do not affect protein kinase activity when the kinase is bound to membranes but do inhibit the solubilized membrane-bound kinase. In the erythrocyte, there is a cytosolic form of the casein kinase which is very similar, having the same molecular weight and substrate specificity as the membrane-bound casein kinase. The cytosolic casein kinase is inhibited by 2,3-diphosphoglycerate but much less so by glycophorin preparations containing phosphoinositol 4,5-bisphosphate. When the sequences of both casein kinases were compared by two-dimensional peptide mapping, it was found that the two kinases were very similar but not identical.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Casein Kinases
  • Chromatography, Affinity
  • Cytosol / enzymology
  • Erythrocyte Membrane / enzymology*
  • Erythrocytes / enzymology
  • Glycophorins / metabolism
  • Humans
  • Kinetics
  • Liposomes
  • Micelles
  • Peptide Mapping
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositols / blood
  • Phosphatidylinositols / pharmacology*
  • Phospholipids / pharmacology
  • Protein Binding
  • Protein Kinases / blood*
  • Protein Kinases / isolation & purification

Substances

  • Glycophorins
  • Liposomes
  • Micelles
  • Phosphatidylinositol 4,5-Diphosphate
  • Phosphatidylinositols
  • Phospholipids
  • Protein Kinases
  • Casein Kinases