Blockade of bombesin receptors with [Leu14-psi(CH2NH)-Leu13]bombesin fails to suppress nutrient-induced CCK release from rat duodenojejunum

Peptides. 1990 Mar-Apr;11(2):255-8. doi: 10.1016/0196-9781(90)90078-j.

Abstract

The present study was undertaken in order to delineate the contribution of enteric bombesin (BBS)-containing nerves in the food-induced release of intestinal cholecystokinin (CCK). For this purpose, the isolated vascularly perfused rat duodenojejunum model was used and the new compound [Leu14-psi(CH2NH)-Leu13]BBS was infused intraarterially at a concentration of 10(-6) M to block the BBS receptors. Vascular infusion of BBS alone (10(-8) M or 10(-9) M) provoked a dose-dependent release of CCK-like immunoreactivity (CCK-LI). The secretion pattern of CCK was biphasic and consisted of a transient peak (300-400% above basal) followed by a sustained response (200-300% above basal). Vascular coinfusion of the BBS analogue with BBS 10(-9) M completely abolished both phases of CCK release while only the second phase of CCK secretion was profoundly reduced upon coadministration of BBS 10(-8) M with the BBS receptor antagonist. Luminal administration of mixed nutrients induced a prompt and well-sustained release of CCK-LI which was unaffected upon arterial infusion of the BBS analogue. These data suggest that the intestinal supply in BBS-producing nerves is not involved in the food-induced release of intestinal CCK in the rat.

MeSH terms

  • Animals
  • Bombesin / analogs & derivatives*
  • Bombesin / metabolism*
  • Bombesin / pharmacology
  • Cholecystokinin / metabolism*
  • Diet
  • Duodenum / innervation
  • Duodenum / metabolism*
  • Jejunum / innervation
  • Jejunum / metabolism*
  • Male
  • Neurons / metabolism
  • Radioimmunoassay
  • Rats
  • Rats, Inbred Strains
  • Receptors, Bombesin
  • Receptors, Neurotransmitter / antagonists & inhibitors*

Substances

  • Receptors, Bombesin
  • Receptors, Neurotransmitter
  • bombesin, Leu(13)-psi-CH2NH-Leu(14)-
  • Cholecystokinin
  • Bombesin