Mechanism and biological significance of the Ha-ras-induced activation of the Na+/H(+)-antiporter

Adv Enzyme Regul. 1990:30:63-74. doi: 10.1016/0065-2571(90)90009-q.

Abstract

Expression of the transforming Ha-ras oncogene in MMTV-LTR transfected NIH 3T3 cells leads to a growth factor independent activation of the Na+/H(+)-antiporter. The activation of the antiporter is insensitive to the protein kinase inhibitor staurosporine and equally expressed in protein kinase C-depleted cells. It is concluded that the Ha-ras induced activation of the antiporter occurs by a protein kinase C-independent mechanism. An inhibition of the Na+/H(+)-antiporter by dimethylamiloride or a reduction of the extracellular [Na+] concentration results in a depression of the bombesin induced release of Ca2+ from intracellular stores. These results are explained by a steep pH-dependence of the Ca2(+)-mobilizing system which exhibits a maximum at pH 7.1 in the system studied here. Stimulation by growth factors of quiescent cells with a resting pH below 7 results in a shift of the cytosolic pH towards the optimum for the Ca2+ release. In agreement with the proposed interrelationship, pHi and [Ca2+]i rise and peak simultaneously after addition of bombesin to G0 arrested cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkaloids / pharmacology
  • Animals
  • Bombesin / pharmacology
  • Calcium / metabolism
  • Carrier Proteins / metabolism*
  • Cell Line
  • Cytosol / metabolism
  • Dexamethasone / pharmacology
  • Genes, ras*
  • Hydrogen-Ion Concentration
  • Kinetics
  • Mammary Tumor Virus, Mouse / genetics
  • Mice
  • Protein Kinase C / antagonists & inhibitors
  • Sodium-Hydrogen Exchangers
  • Staurosporine
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transfection

Substances

  • Alkaloids
  • Carrier Proteins
  • Sodium-Hydrogen Exchangers
  • Dexamethasone
  • Protein Kinase C
  • Staurosporine
  • Tetradecanoylphorbol Acetate
  • Bombesin
  • Calcium